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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
Athersys, Inc.
Curated by
ChEMBL
Ligand
BDBM50162903
(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)
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copy InChI
Affinity Data
Ki: 13nM
Assay Description:
Inhibitory activity of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calcium
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20P0ZHT
PubMed
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
Athersys, Inc.
Curated by
ChEMBL
Ligand
BDBM50162903
(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)
copy SMILES
copy InChI
Affinity Data
Ki: >2.00E+4nM
Assay Description:
Inhibitory activity of the compound for binding of PGD-2 in hTP binding assay using HEK293 cell membranes
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20P0ZHT
PubMed
Target
Prostaglandin D2 receptor 2
(Homo sapiens (Human))
Athersys, Inc.
Curated by
ChEMBL
Ligand
BDBM50162903
(CHEMBL359855 | [6-(4-Fluoro-benzenesulfonylamino)-...)
copy SMILES
copy InChI
Affinity Data
IC50: 9.70nM
Assay Description:
Inhibitory concentration of the compound for PGD2-mediated receptor activation in a fluorescence assay that measures changes in intracellular calcium
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20P0ZHT
PubMed