Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetProtein kinase C delta type(Homo sapiens (Human))
National Institutes of Health

LigandPNGBDBM92596(Sapintoxin D)copy SMILEScopy InChI
Affinity DataKi:  0.140nM ΔG°:  -54.9kJ/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9NQ6PubMed
TargetSerine/threonine-protein kinase MRCK alpha(Homo sapiens (Human))
National Institutes of Health

LigandPNGBDBM92596(Sapintoxin D)copy SMILEScopy InChI
Affinity DataKi:  5.90nM ΔG°:  -45.9kJ/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9NQ6PubMed
TargetSerine/threonine-protein kinase MRCK beta(Homo sapiens (Human))
National Institutes of Health

LigandPNGBDBM92596(Sapintoxin D)copy SMILEScopy InChI
Affinity DataKi:  12.6nM ΔG°:  -44.0kJ/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9NQ6PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
National Institutes of Health

LigandPNGBDBM92596(Sapintoxin D)copy SMILEScopy InChI
Affinity DataKi:  18.2nM ΔG°:  -43.1kJ/molepH: 7.4 T: 2°CAssay Description:[3H]PDBu binding to the C1 domains of MRCK alpha/beta and PKC alpha/delta was measured using the polyethylene glycol precipitation assay.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9NQ6PubMed