Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50468281(CHEMBL4294862)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2C9TPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50468281(CHEMBL4294862)copy SMILEScopy InChI
Affinity DataIC50: 80nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2C9TPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50468281(CHEMBL4294862)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2C9TPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50468281(CHEMBL4294862)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2C9TPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50468281(CHEMBL4294862)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K2C9TPubMed