Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre
Curated by
ChEMBL
Ligand
BDBM50099953
(CHEMBL3319604)
copy SMILES
copy InChI
Affinity Data
IC50: 95nM
Assay Description:
Inhibition of proteasome subunit beta-1i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BR8TZT
PubMed
Target
Proteasome subunit beta type-9
(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre
Curated by
ChEMBL
Ligand
BDBM50099953
(CHEMBL3319604)
copy SMILES
copy InChI
Affinity Data
IC50: 130nM
Assay Description:
Inhibition of proteasome subunit beta-1i in human RPMI8226 cells using BODIPY-NC001 by fluorescent densitometry
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BR8TZT
PubMed
Target
Proteasome subunit beta type-10
(Homo sapiens (Human))
Leiden Institute of Chemistry and Netherlands Proteomics Centre
Curated by
ChEMBL
Ligand
BDBM50099953
(CHEMBL3319604)
copy SMILES
copy InChI
Affinity Data
IC50: 1.00E+5nM
Assay Description:
Inhibition of proteasome subunit beta-2i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2BR8TZT
PubMed