Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 105 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataKi:  0.0460nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC1 receptor expressed in BHK570 cells after 90 mins in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataKi:  0.300nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from MC4 receptor after 2 hrs by gamma counting in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataKi:  0.480nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor human MC5 expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataKi:  0.780nMAssay Description:Displacement of [125I]-NAD-alpha-MSH from human recombinant MC3 receptor expressed in BHK570 cells after 1 hr in presence of ovalbuminMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDP-a-MSH from human recombinant MC4 receptor expressed in CHO cells measured after 120 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CF9S3SPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.150nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human recombinant MC4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J67JS7PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.290nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 1 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.310nMAssay Description:Displacement of 125I-NDP-MSH from mouse MC1R expressed in HEK293 cells incubated for 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.400nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 4 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 0.890nMAssay Description:Binding affinity for Human Melanocortin 5 receptor expressed in L-cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 1.10nMAssay Description:Displacement of 125I-NDP-MSH from mouse MC4R expressed in HEK293 cells incubated for 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]-NDP-MSH from mouse MC4R expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 5 receptor expressed in HEK293 cells; N = 4More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMAssay Description:Binding affinity for Human Melanocortin 3 receptor expressed in L-cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Inhibition of [125I]NDP-MSH binding to Melanocortin 3 receptor expressed in HEK293 cells; (N = 4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 3.30nMAssay Description:Binding affinity for Human Melanocortin 4 receptor expressed in L-cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 4.20nMAssay Description:Displacement of 125I-NDP-MSH from mouse MC3R expressed in HEK293 cells incubated for 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]-NDP-MSH from mouse MC3R expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 8.20nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 3 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-NDP-MSH from human melanocortin receptor 4 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 14nMAssay Description:Displacement of [I125]-NDP-MSH from wild type human melanocortin-4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ347JPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataIC50: 140nMAssay Description:Displacement of [125I]-NDP-MSH from mouse melanocortin receptor 5 expressed in HEK293 cell mebranes incubated for 1 hr by automatic gamma counting me...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0880nMAssay Description:Agonist activity at mouse melanocortin-1 receptor expressed in HEK293 cells co-transfected with CRE/beta-galactosidase reporter gene assessed as stim...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ347JPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at mouse melanocortin-3 receptor expressed in HEK293 cells co-transfected with CRE/beta-galactosidase reporter gene assessed as stim...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ347JPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse melanocortin-4 receptor expressed in HEK293 cells co-transfected with CRE/beta-galactosidase reporter gene assessed as stim...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ347JPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at mouse melanocortin-5 receptor expressed in HEK293 cells co-transfected with CRE/beta-galactosidase reporter gene assessed as stim...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ347JPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0180nMAssay Description:Agonist activity at mouse melanocortin 1 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB537CPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at mouse melanocortin 5 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB537CPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at mouse melanocortin 3 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB537CPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at mouse melanocortin 4 receptor expressed in HEK293 cells after 48 hrs by cAMP based beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FB537CPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0460nMAssay Description:Maximal agonist response of mouse melanocortin 1 receptor (MC1R)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP75PKPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.290nMAssay Description:Effective concentration for maximum agonist response towards mouse melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP75PKPubMed
TargetMelanocortin receptor 3(Rattus norvegicus)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.100nMAssay Description:Maximal agonist response at rat melanocortin 3 receptor (MC3R)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP75PKPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0640nMAssay Description:Maximum agonist response for mouse melanocortin 5 receptor (MC5R)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP75PKPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Effective concentration for intracellular cAMP accumulation in human melanocortin 3 receptor expressing HEK 293 cells; (N = 4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Effective concentration for intracellular cAMP accumulation in human melanocortin 5 receptor expressing HEK 293 cells; (N = 4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Effective concentration for intracellular cAMP accumulation in human melanocortin 4 receptor expressing HEK 293 cells; (N = 4)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XD12F5PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.240nMAssay Description:Effective concentration required for intracellular cAMP accumulation against Melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Effective concentration required for intracellular cAMP accumulation by Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.230nMAssay Description:Effective concentration required for intracellular cAMP accumulation by Melanocortin 5 receptorMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2P55P7VPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0170nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 4 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.130nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0230nMAssay Description:Effective concentration required for the biological activity against human Melanocortin 1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JW8FM1PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human recombinant MC4 receptor expressed in BHK570 cells assessed as induction of cMAP accumulation in presence of 0.1% human ser...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN464PPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0920nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.810nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation incubated for 2 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation incubated for 2 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.460nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation incubated for 2 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation incubated for 2 hrs by alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R2139SPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.390nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as induction of cAMP accumulation after 2 hrs by alpha screen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24170J1PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0700nMAssay Description:Displacement of Eu-NDP-MSH from human MC1R expressed in HEK293T cells after 2 hrs by DELFIA methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.870nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in cAMP production incubated for 2 hrs by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CV4M69PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN47H1PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0210nMAssay Description:Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN47H1PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN47H1PubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as increase in cAMP accumulation after 2 hrs by AlphaScreen assa...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN47H1PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells incubated for 2 hrs by AlphaScreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QHMPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Inverse agonist activity at mouse MC5R expressed in HEK293 cells incubated for 2 hrs by AlphaScreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X63QHMPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk A/S

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ3535PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25142KGPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.279nMAssay Description:Agonist activity at mouse MC4R expressed in HEK293 cells co-expressing CRE/beta-galactosidase reporter gene after 6 hrs by beta-galactosidase cAMP as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2SWGPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.414nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells co-expressing CRE/beta-galactosidase reporter gene after 6 hrs by beta-galactosidase cAMP as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2SWGPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0510nMAssay Description:Full agonist activity at mouse MC1R expressed in HEK293 cells co-expressing CRE/beta-galactosidase reporter gene after 6 hrs by beta-galactosidase cA...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2SWGPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  2nMAssay Description:Full agonist activity at mouse MC5R expressed in HEK293 cells co-expressing CRE/beta-galactosidase reporter gene after 6 hrs by beta-galactosidase cA...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2SWGPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0120nMAssay Description:Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QTBPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QTBPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QTBPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QV3QTBPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.00600nMAssay Description:Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301KKPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301KKPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301KKPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of cAMP accumulation incubated for 2 hrs by cAMP ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301KKPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0100nMAssay Description:Agonist activity at mouse MC1R by alphascreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ36C5PubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at mouse MC3R by alphascreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ36C5PubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at mouse MC4R by alphascreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ36C5PubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at mouse MC5R by alphascreen cAMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ36C5PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0120nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as induction of cAMP level at 100 uM incubated for 2 hr by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR231GPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0740nMAssay Description:Agonist activity at mouse MC3R expressed in HEK293 cells assessed as induction of cAMP level incubated for 2 hr by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR231GPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as induction of cAMP level at 100 uM incubated for 2 hr by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR231GPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at mouse melanocortin receptor 1 expressed in HEK293 cells assessed as stimulation of intracellular cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S0NPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.360nMAssay Description:Agonist activity at mouse melanocortin receptor 3 expressed in HEK293 cells assessed as stimulation of intracellular cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S0NPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as stimulation of intracellular cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S0NPubMed
TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)copy SMILEScopy InChI
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse melanocortin receptor 5 expressed in HEK293 cells assessed as stimulation of intracellular cAMP accumulation incubated for ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5S0NPubMed
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