Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)copy SMILEScopy InChI
Affinity DataEC50:  1.90nMAssay Description:Activity at mouse MC5R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)copy SMILEScopy InChI
Affinity DataEC50:  0.240nMAssay Description:Activity at mouse MC1R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocortin receptor 3(Mus musculus)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)copy SMILEScopy InChI
Affinity DataEC50:  1.90nMAssay Description:Activity at mouse MC3R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed
TargetMelanocortin receptor 4(Mus musculus)
University of Cergy-Pontoise

Curated by ChEMBL
LigandPNGBDBM50031494(CHEMBL3358537)copy SMILEScopy InChI
Affinity DataEC50:  0.810nMAssay Description:Activity at mouse MC4R expressed in HEK293 cells assessed as cAMP accumulation by CRE/beta-galactosidase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21G0NVTPubMed