Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
Ki: 9nM ΔG°: -47.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
Ki: 1.00E+4nM ΔG°: -29.7kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
Ki: 1.00E+4nM ΔG°: -29.7kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
BDBM250665(US9447148, 9.34 | US9447148, 9.47)copy SMILES
EC50: 4nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair