Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126093(CHEMBL386871 | MT-II cyclic peptide derivative)copy SMILEScopy InChI
Affinity DataEC50:  45nMAssay Description:Agonist activity at human melanocortin receptor (hMC4R).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J994CPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50126093(CHEMBL386871 | MT-II cyclic peptide derivative)copy SMILEScopy InChI
Affinity DataEC50:  480nMAssay Description:Agonist activity at human melanocortin receptor (hMC1R).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21J994CPubMed