Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetOxytocin receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50314512(5-(2,3-dimethylphenyl)-N-ethyl-N-(6-methoxypyridin...)copy SMILEScopy InChI
Affinity DataKi:  25nMAssay Description:Antagonist activity at human cloned OT receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XMSPubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50314512(5-(2,3-dimethylphenyl)-N-ethyl-N-(6-methoxypyridin...)copy SMILEScopy InChI
Affinity DataKi:  2.83E+3nMAssay Description:Antagonist activity at human cloned vasopressin V2 receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XMSPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
Pfizer Global Research and Development

Curated by ChEMBL
LigandPNGBDBM50314512(5-(2,3-dimethylphenyl)-N-ethyl-N-(6-methoxypyridin...)copy SMILEScopy InChI
Affinity DataKi:  4.72E+5nMAssay Description:Antagonist activity at human cloned vasopressin V1A receptor by cell based beta-lactamase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X34XMSPubMed