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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by
ChEMBL
Ligand
BDBM50397206
(CHEMBL2172289)
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Affinity Data
Ki: 5.69nM
Assay Description:
Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 mins
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q28G8MT5
PubMed
Target
Oxytocin receptor
(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by
ChEMBL
Ligand
BDBM50397206
(CHEMBL2172289)
copy SMILES
copy InChI
Affinity Data
Ki: 184nM
Assay Description:
Displacement of [3H]-AVP from human oxytocin receptor expressed in CHO cells after 30 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q28G8MT5
PubMed
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by
ChEMBL
Ligand
BDBM50397206
(CHEMBL2172289)
copy SMILES
copy InChI
Affinity Data
Ki: 621nM
Assay Description:
Displacement of [3H]-AVP from human vasopressin V1a receptor expressed in CHO cells after 30 mins
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q28G8MT5
PubMed
Target
Vasopressin V1b receptor
(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by
ChEMBL
Ligand
BDBM50397206
(CHEMBL2172289)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Displacement of [3H]-AVP from human vasopressin V1b receptor expressed in CHO cells after 30 mins
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q28G8MT5
PubMed
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
UMR7200 CNRS/Universit£ de Strasbourg
Curated by
ChEMBL
Ligand
BDBM50397206
(CHEMBL2172289)
copy SMILES
copy InChI
Affinity Data
Kd: 1.38nM
Assay Description:
Binding affinity to SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells after 1 hr by TR-FRET assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q28G8MT5
PubMed