Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 6(Homo sapiens (Human))
Universit£t Leipzig

Curated by ChEMBL
LigandPNGBDBM50299473(CHEMBL577248 | Ethyl 2-amino-5-(4-methoxyphenyl)-4...)copy SMILEScopy InChI
Affinity DataIC50: 8.60E+3nMAssay Description:Antagonist activity at human recombinant GluR6 expressed in HEK cells coexpressing aequorine assessed as inhibition of glutamate-induced Ca2+ influx ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4QVFPubMed