Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
GALDERMA RESEARCH & DEVELOPMENT

US Patent
LigandPNGBDBM323184(N-[(S)-2-(3-ethoxy-3-o-tolylazetidin-1-yl)-1-(4-me...)copy SMILEScopy InChI
Affinity DataEC50:  1.50E+4nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21Z46H9US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
GALDERMA RESEARCH & DEVELOPMENT

US Patent
LigandPNGBDBM323184(N-[(S)-2-(3-ethoxy-3-o-tolylazetidin-1-yl)-1-(4-me...)copy SMILEScopy InChI
Affinity DataEC50:  2.00E+3nMAssay Description:In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21Z46H9US Patent