Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetRelaxin-3 receptor 2(Homo sapiens (Human))TBA
LigandPNGBDBM50581020(CHEMBL5094669)copy SMILES
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human RXFP4 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5MJPPubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM50581020(CHEMBL5094669)copy SMILES
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human RXFP3 expressed in human CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 1.5 hrs ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5MJPPubMed