Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM572236((6S)-1-methyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)copy SMILES
BDBM572236((6S)-1-methyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)copy SMILES
Ki: 0.0280nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572236((6S)-1-methyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)copy SMILES
Ki: 4.19nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572236((6S)-1-methyl-8-(3-pyrimidin-4-yl-1H-pyrrolo[2,3- ...)copy SMILES
Ki: 20.6nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair