Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 32 hits in this display
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
IC50: 1.34E+3nMAssay Description:Inhibition of N-[3',6'-dihydroxy-3-oxo-3H-spiro(2-benzofuran-1,9'-xanthen)-5-yl]-N'-[2-(4-{4-[N-(2-chloro-6-methylphenyl)-5-carboxamido]-thiazol-2-yl...More data for this Ligand-Target Pair
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
IC50: 4.94E+3nMAssay Description:Inhibition of human full length PKMYT1 expressed in HEK293 cells using EFS (247 to 259 residues) as substrate after 1 hr by fluorescence polarization...More data for this Ligand-Target Pair
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI
Kd: 324nMAssay Description:Binding affinity to recombinant human N-terminal His6-tagged Myt1 kinase domain (75 to 361 residues) by isothermal titration calorimetryMore data for this Ligand-Target Pair
BDBM50240826(AZD-1775 | MK-1775 | US11124518, Example AZD1775 |...)copy SMILEScopy InChI