Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 43nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 84nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 84nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 736nM ΔG°: -36.4kJ/molepH: 7.4 T: 2°CAssay Description:The assay was performed at 37 °C in HEPES buffer (100 mM, with 10% glycerol, pH 7.4) in the presence of 10 uM L-arginine. Also included were 100 ...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 748nM ΔG°: -36.4kJ/molepH: 7.4 T: 2°CAssay Description:The assay was performed at 37 °C in HEPES buffer (100 mM, with 10% glycerol, pH 7.4) in the presence of 10 uM L-arginine. Also included were 100 ...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 1.42E+4nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: >3.00E+4nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI
Ki: 7.30E+4nMAssay Description:Enzyme inhibition was evaluated by measuring NO production with the hemoglobin capture assay, which was performed with purified NOSs in 96-well plate...More data for this Ligand-Target Pair
BDBM190665(US10759791, Compound 14g | nNOS inhibitor, 3)copy SMILEScopy InChI