Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetMelanocortin receptor 4(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataKi:  1.10nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataKi:  2nMAssay Description:Binding affinity to human MC1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataKi:  3.30nMAssay Description:Binding affinity to human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataEC50:  0.370nMAssay Description:Agonist activity at human MC1RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataEC50:  0.340nMAssay Description:Agonist activity at human MC4RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189025((S)-2-acetamido-N1-((R)-3-(4-fluorophenyl)-1-((S)-...)copy SMILEScopy InChI
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human MC3RMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66KDFPubMed