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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
Otsuka Pharmaceutical Co., Ltd
Ligand
BDBM35715
(benzazepine derivative, 13a)
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copy InChI
Affinity Data
IC50: 7nM
pH: 7.4 T: 2°C
Assay Description:
After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W957JR
PubMed
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
Otsuka Pharmaceutical Co., Ltd
Ligand
BDBM35715
(benzazepine derivative, 13a)
copy SMILES
copy InChI
Affinity Data
IC50: 64nM
pH: 7.4 T: 2°C
Assay Description:
After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W957JR
PubMed