Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 8 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataKi:  328nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC1 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataKi:  403nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataKi:  1.53E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC5 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataKi:  4.53E+3nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC5 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataEC50:  12nMAssay Description:Agonist activity at human MC1 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataEC50:  697nMAssay Description:Agonist activity at human MC4 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed
TargetMelanocortin receptor 3(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50337289(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human MC3 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9PPVPubMed