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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
8
hits in this display
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
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Affinity Data
Ki: 328nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human MC1 receptor expressed in BHK cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
Ki: 403nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human MC4 receptor expressed in BHK cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
Ki: 1.53E+3nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human MC5 receptor expressed in BHK cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
Ki: 4.53E+3nM
Assay Description:
Displacement of [125I]NDP-alpha-MSH from human MC3 receptor expressed in BHK cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Agonist activity at human MC5 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
EC50: 12nM
Assay Description:
Agonist activity at human MC1 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
EC50: 697nM
Assay Description:
Agonist activity at human MC4 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Novo Nordisk
Curated by
ChEMBL
Ligand
BDBM50337289
(CHEMBL1682208 | N-[(13S)-15-{3-[4-(3-aminopropyl)p...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Agonist activity at human MC3 receptor expressed in BHK cells assessed as stimulation of agonist-induced cAMP accumulation
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q20R9PPV
PubMed