Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  1.84E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  1.15E+4nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE

US Patent
LigandPNGBDBM196907(US9212196, Derivative 3)copy SMILEScopy InChI
Affinity DataEC50:  4.70E+3nMAssay Description:Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q28G8JJRUS Patent