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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Metabotropic glutamate receptor 4
(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE
US Patent
Ligand
BDBM196907
(US9212196, Derivative 3)
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copy InChI
Affinity Data
EC50: 100nM
Assay Description:
Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q28G8JJR
US Patent
Target
Metabotropic glutamate receptor 8
(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE
US Patent
Ligand
BDBM196907
(US9212196, Derivative 3)
copy SMILES
copy InChI
Affinity Data
EC50: 1.84E+4nM
Assay Description:
Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q28G8JJR
US Patent
Target
Metabotropic glutamate receptor 7
(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE
US Patent
Ligand
BDBM196907
(US9212196, Derivative 3)
copy SMILES
copy InChI
Affinity Data
EC50: 1.15E+4nM
Assay Description:
Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q28G8JJR
US Patent
Target
Metabotropic glutamate receptor 6
(Rattus norvegicus (Rat))
UNIVERSITE PARIS DESCARTES; UNIVERSITE D'AUVERGNE
US Patent
Ligand
BDBM196907
(US9212196, Derivative 3)
copy SMILES
copy InChI
Affinity Data
EC50: 4.70E+3nM
Assay Description:
Metabotropic glutamate receptors were transiently transfected in HEK293 cells by electroporation as described elsewhere (Brabet I. et al., 1998) and ...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q28G8JJR
US Patent