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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Melanocortin receptor 4
(Homo sapiens (Human))
GALDERMA RESEARCH & DEVELOPMENT
US Patent
Ligand
BDBM323199
(N-[(R)-2-(3-cyclopropylmethoxy-3-phenylazetidin-1-...)
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copy InChI
Affinity Data
EC50: 8.00E+3nM
Assay Description:
In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q21Z46H9
US Patent
Target
Melanocyte-stimulating hormone receptor
(Homo sapiens (Human))
GALDERMA RESEARCH & DEVELOPMENT
US Patent
Ligand
BDBM323199
(N-[(R)-2-(3-cyclopropylmethoxy-3-phenylazetidin-1-...)
copy SMILES
copy InChI
Affinity Data
EC50: 1.00E+3nM
Assay Description:
In the presence of an activator (agonist), the melanocortin receptor will activate the cAMP pathway which, via the CRE-Luc vector, will result in the...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q21Z46H9
US Patent