Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Amgen

LigandPNGBDBM365040(4-(3-(3-fluoro-4- methoxybenzyl)-4,5-dihydro- 3H-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NV9MJ5US Patent
TargetMitogen-activated protein kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM365040(4-(3-(3-fluoro-4- methoxybenzyl)-4,5-dihydro- 3H-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KP85BCUS Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))
Amgen

LigandPNGBDBM365040(4-(3-(3-fluoro-4- methoxybenzyl)-4,5-dihydro- 3H-1...)copy SMILEScopy InChI
Affinity DataIC50: 0.311nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q23X88ZRUS Patent