Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetOxytocin receptor(Homo sapiens (Human))
GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413724(CHEMBL459073)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Antagonist activity at human recombinant oxytocin receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29Z5FPubMed
TargetVasopressin V1a receptor(Homo sapiens (Human))
GlaxoSmithKline Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50413724(CHEMBL459073)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human recombinant vasopressin V1a receptor expressed in CHO cells by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N29Z5FPubMed