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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Oxytocin receptor
(Homo sapiens (Human))
Pfizer Global Research and Development
Curated by
ChEMBL
Ligand
BDBM50305525
(5-(3-(3-(5-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
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Affinity Data
Ki: 40nM
Assay Description:
Antagonist activity at human cloned oxytocin receptor by cell based beta lactamase assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MS3SWF
PubMed
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
Pfizer Global Research and Development
Curated by
ChEMBL
Ligand
BDBM50305525
(5-(3-(3-(5-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
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copy InChI
Affinity Data
Ki: 1.68E+3nM
Assay Description:
Antagonist activity at human cloned vasopressin V1a receptor by cell based beta lactamase assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MS3SWF
PubMed
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
Pfizer Global Research and Development
Curated by
ChEMBL
Ligand
BDBM50305525
(5-(3-(3-(5-fluoro-2-methylphenoxy)azetidin-1-yl)-5...)
copy SMILES
copy InChI
Affinity Data
Ki: 2.77E+3nM
Assay Description:
Antagonist activity at human cloned vasopressin V2 receptor by cell based beta lactamase assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MS3SWF
PubMed