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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
9
hits in this display
Target
Prostaglandin E2 receptor EP4 subtype
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
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Affinity Data
Ki: 0.790nM
Assay Description:
Binding affinity to human EP4 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin E2 receptor EP4 subtype
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 1.60nM
Assay Description:
Binding affinity to human EP4 receptor expressed in HEK293 cells in presence of 10% human serum
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 39nM
Assay Description:
Binding affinity to human TP receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin D2 receptor
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
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copy InChI
Affinity Data
Ki: 53nM
Assay Description:
Binding affinity to human DP receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin E2 receptor EP2 subtype
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 300nM
Assay Description:
Binding affinity to human EP2 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin F2-alpha receptor
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 340nM
Assay Description:
Binding affinity to human FP receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostacyclin receptor
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 2.00E+3nM
Assay Description:
Binding affinity to human IP receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin E2 receptor EP3 subtype
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: 2.70E+3nM
Assay Description:
Binding affinity to human EP3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed
Target
Prostaglandin E2 receptor EP1 subtype
(Homo sapiens (Human))
Merck Frosst Centre for Therapeutic Research
Curated by
ChEMBL
Ligand
BDBM50372058
(CHEMBL404199)
copy SMILES
copy InChI
Affinity Data
Ki: >9.00E+3nM
Assay Description:
Binding affinity to human EP1 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2J96770
PubMed