Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetSomatostatin receptor type 1(RAT)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50423302(CHEMBL248715)copy SMILEScopy InChI
Affinity DataKd:  1.20nMAssay Description:Displacement of [125I]SRIF14 from sst1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP7675PubMed
TargetSomatostatin receptor type 1(RAT)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50423302(CHEMBL248715)copy SMILEScopy InChI
Affinity DataKd:  1.20nMAssay Description:Displacement of [125I]SRIF14 from rat sst1 receptor from rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6FHFPubMed
TargetSomatostatin receptor type 2(RAT)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50423302(CHEMBL248715)copy SMILEScopy InChI
Affinity DataKd:  5.75E+3nMAssay Description:Displacement of [125I]SRIF14 from rat sst2 receptor from rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2SX6FHFPubMed
TargetSomatostatin receptor type 2(RAT)
Novartis Institutes for BioMedical Research

Curated by ChEMBL
LigandPNGBDBM50423302(CHEMBL248715)copy SMILEScopy InChI
Affinity DataKd:  5.75E+3nMAssay Description:Displacement of [125I]SRIF14 from sst2 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XP7675PubMed