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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
142
hits in this display
Target
Rho-associated protein kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 2nM
Assay Description:
Inhibition of ROCK1 (6 to 553 residues) (unknown origin) using Lys-Lys-Arg-Asn-Arg-Thr-Leu-Ser-Val as substrate in presence of ATP by spectrophotomet...
More data for this Ligand-Target Pair
Target Info
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Article
BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
PDB
3D Structure (crystal)
Target
Rho-associated protein kinase 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: <4nM
Assay Description:
Inhibition of ROCK2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Article
BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Rho-associated protein kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
copy SMILES
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Affinity Data
Ki: 6nM
Assay Description:
Inhibition of ROCK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Article
BindingDB Entry DOI:
10.7270/Q2805665
PubMed
PDB
3D Structure (crystal)
Target
Serine/threonine-protein kinase N2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 77nM
Assay Description:
Inhibition of PRK2 (unknown origin)
More data for this Ligand-Target Pair
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NCI pathway
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ribosomal protein S6 kinase alpha-5
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 94nM
Assay Description:
Inhibition of MSK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ribosomal protein S6 kinase alpha-1/alpha-2/alpha-3/alpha-4/alpha-5/alpha-6/beta-1/beta-2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 100nM
Assay Description:
Inhibition of p70S6K (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Article
BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Citron Rho-interacting kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 160nM
Assay Description:
Inhibition of CIT (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C gamma type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 210nM
Assay Description:
Inhibition of PKCgamma (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Receptor-type tyrosine-protein kinase FLT3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 250nM
Assay Description:
Inhibition of FLT3 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase JAK3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 280nM
Assay Description:
Inhibition of JAK3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C theta type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 290nM
Assay Description:
Inhibition of PKCtheta (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase JAK2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 400nM
Assay Description:
Inhibition of JAK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 400nM
Assay Description:
Inhibition of GSK3beta (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C epsilon type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 690nM
Assay Description:
Inhibition of PKCepsilon (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 890nM
Assay Description:
Inhibition of Erk2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ribosomal protein S6 kinase alpha-2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 940nM
Assay Description:
Inhibition of RSK3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase kinase kinase kinase 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Inhibition of MAP4K4 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 1A
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 1.00E+3nM
Assay Description:
Inhibition of DYRK1A (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase D2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Inhibition of PRKD2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
PAS domain-containing serine/threonine-protein kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Inhibition of PASK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity mitogen-activated protein kinase kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Inhibition of MEK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Misshapen-like kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+3nM
Assay Description:
Inhibition of MINK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Cyclin-dependent kinase 5 activator 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 1.30E+3nM
Assay Description:
Inhibition of CDK5/p35 (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Cyclin-A2/Cyclin-dependent kinase 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 1.50E+3nM
Assay Description:
Inhibition of CDK2/CycA (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Interleukin-1 receptor-associated kinase 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 1.90E+3nM
Assay Description:
Inhibition of IRAK4 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase ZAP-70
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of ZAP70 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of IGF1R (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Fibroblast growth factor receptor 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FGFR2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 13
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of p38delta (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ribosomal protein S6 kinase alpha-1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of RSK1 (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity protein kinase CLK3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CLK3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase PAK 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PAK3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PHKgamma2 (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase pim-2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of Pim2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Calcium/calmodulin-dependent protein kinase type II subunit beta
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CamK2B (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Calcium/calmodulin-dependent protein kinase type II subunit beta
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CamK2 (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Chk1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CheK1 (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Chk2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CheK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase CSK
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CSK (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ephrin type-B receptor 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of EphB2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Vascular endothelial growth factor receptor 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FLT4 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Fyn
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FYN (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase MARK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MARK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase D3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PRKD3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Sgk2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of SGK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Testis-specific serine/threonine-protein kinase 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of TSSK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Yes
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of YES (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity mitogen-activated protein kinase kinase 7
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MKK7 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 12
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of p38gamma (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase ABL1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of Abl1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Death-associated protein kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of DAPK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Mer
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MER (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Nek1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of NEK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase PAK 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PAK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity mitogen-activated protein kinase kinase 6
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MKK6 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MST1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Nek2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of NEK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase PAK 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PAK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase pim-1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of Pim1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C beta type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PKCbeta1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase D1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PRKD1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein-tyrosine kinase 2-beta
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of PYK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Macrophage-stimulating protein receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of RON (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Proto-oncogene tyrosine-protein kinase ROS
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of ROS (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ribosomal protein S6 kinase alpha-3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of RSK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Sgk1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of SGK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Sgk3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of SGK3 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase TBK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of TBK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Angiopoietin-1 receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of TIE2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase receptor TYRO3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of TYRO3 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Calcium/calmodulin-dependent protein kinase type 1D
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of Camk1D (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Calcium/calmodulin-dependent protein kinase type II subunit alpha
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of Camk2A (unknown origin)
More data for this Ligand-Target Pair
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Calcium/calmodulin-dependent protein kinase type IV
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CamK4 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Cyclin-dependent kinase/G2/mitotic-specific cyclin- 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CDK1/CycB (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Casein kinase I isoform alpha
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of CK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase DCLK2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of DCAMKL2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ephrin type-B receptor 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of EphB4 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Fes/Fps
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FES (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FGFR1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FGFR3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FLT1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Macrophage colony-stimulating factor 1 receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FMS (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase HCK
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of HCK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Inhibitor of nuclear factor kappa-B kinase subunit alpha
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of IKKalpha (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Insulin receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of INSR (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 8
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of JNK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of KIT (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of LCK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of LYN (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
MAP kinase-activated protein kinase 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of MAPKAPK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Proto-oncogene tyrosine-protein kinase receptor Ret
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Ki: >2.00E+3nM
Assay Description:
Inhibition of RET (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Dual specificity tyrosine-phosphorylation-regulated kinase 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of DYRK2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Fer
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FER (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Fibroblast growth factor receptor 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of FGFR4 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C beta type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 2.09E+3nM
Assay Description:
Inhibition of PKCbeta2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Interleukin-1 receptor-associated kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 2.20E+3nM
Assay Description:
Inhibition of IRAK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase kinase kinase 7
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: 2.70E+3nM
Assay Description:
Inhibition of TAK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >2.90E+3nM
Assay Description:
Inhibition of Erk1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of MET (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of PI3Kgamma (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase kinase kinase 8
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Ki: >4.00E+3nM
Assay Description:
Inhibition of COT (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Ki: >4.00E+3nM
Assay Description:
Inhibition of SRC (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of p38alpha (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 10
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of JNK3 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase SYK
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of SYK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >4.00E+3nM
Assay Description:
Inhibition of KDR (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase Sgk1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Ki: >5.00E+3nM
Assay Description:
Inhibition of SGK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
MAP/microtubule affinity-regulating kinase 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Ki: >5.00E+3nM
Assay Description:
Inhibition of cTak1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase TBK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of NAK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase kinase kinase 14
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of NIK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Protein kinase C iota type
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of PKCiota (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Sphingosine kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of SphK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
RAC-alpha serine/threonine-protein kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Akt1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Aurora kinase A
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of AurA (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Cytoplasmic tyrosine-protein kinase BMX
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of BMX (unknown origin)
More data for this Ligand-Target Pair
Target Info
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MMDB
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase DCLK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of DCLK1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
DNA-dependent protein kinase catalytic subunit
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of DNAPK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ephrin type-A receptor 4
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of EphA4 (unknown origin)
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MMDB
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of FAK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Platelet-derived growth factor receptor alpha
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of PDGFRalpha (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
MAP kinase-activated protein kinase 5
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of PRAK (unknown origin)
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Target Info
NCI pathway
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Mitogen-activated protein kinase 11
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of p38beta (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase 3
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of MST2 (unknown origin)
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MMDB
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Aurora kinase B
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of AurB (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
RAC-gamma serine/threonine-protein kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Akt3 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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MMDB
NCI pathway
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
RAF proto-oncogene serine/threonine-protein kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of RAFc (unknown origin)
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Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of PLK1 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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Article
BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of IKKbeta (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase BTK
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Btk (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase BRSK1
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Brsk1 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Choline kinase alpha
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of ChoK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Ceramide kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of CerK (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Aurora kinase C
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of AurC (unknown origin)
More data for this Ligand-Target Pair
Target Info
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NCI pathway
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase BRSK2
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Brsk2 (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
RAC-beta serine/threonine-protein kinase
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Akt2 (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Serine/threonine-protein kinase ATR
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of ATR (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase ITK/TSK
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of ITK (unknown origin)
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Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of EGFR (unknown origin)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
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Article
BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Tyrosine-protein kinase Blk
(Homo sapiens (Human))
Vertex Pharmaceuticals Inc
Curated by
ChEMBL
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of Blk (unknown origin)
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Cytochrome P450 3A4
(Homo sapiens (Human))
TBA
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
IC50: 8.30E+3nM
Assay Description:
Inhibition of CYP3A4 (unknown origin)
More data for this Ligand-Target Pair
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Article
BindingDB Entry DOI:
10.7270/Q2805665
PubMed
Target
Cytochrome P450 3A4
(Homo sapiens (Human))
TBA
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
IC50: 8.30E+3nM
Assay Description:
Inhibition of CYP3A4 (unknown origin)
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2ZC85HX
PubMed
Target
Potassium voltage-gated channel subfamily H member 2
(Homo sapiens (Human))
TBA
Ligand
BDBM50463479
(CHEMBL4249925)
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Affinity Data
IC50: 3.00E+4nM
Assay Description:
Inhibition of human ERG
More data for this Ligand-Target Pair
Target Info
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BindingDB Entry DOI:
10.7270/Q2805665
PubMed
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