Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetNitric oxide synthase, brain(Homo sapiens (Human))
NeurAxon, Inc.

US Patent
LigandPNGBDBM106710(CHEMBL1957357 | US8586620, 75)copy SMILEScopy InChI
Affinity DataIC50: 2.25E+3nMAssay Description:Enzyme assay using recombinant human inducible NOS (iNOS), human endothelial constitutive NOS (eNOS) or human neuronal constitutive NOS (nNOS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348J0KUS Patent
TargetNitric oxide synthase, brain(Homo sapiens (Human))
NeurAxon, Inc.

US Patent
LigandPNGBDBM106710(CHEMBL1957357 | US8586620, 75)copy SMILEScopy InChI
Affinity DataIC50: 2.25E+3nMAssay Description:Inhibition of human nNOS expressed in baculovirus infected insect Sf9 cells assessed as conversion of [3H]-L-arginine to [3H]-L-citrullineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52Q3NPubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
NeurAxon Inc.

Curated by ChEMBL
LigandPNGBDBM106710(CHEMBL1957357 | US8586620, 75)copy SMILEScopy InChI
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of human iNOS expressed in baculovirus infected insect Sf9 cells assessed as conversion of [3H]-L-arginine to [3H]-L-citrullineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52Q3NPubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
NeurAxon Inc.

Curated by ChEMBL
LigandPNGBDBM106710(CHEMBL1957357 | US8586620, 75)copy SMILEScopy InChI
Affinity DataIC50: 3.61E+4nMAssay Description:Inhibition of human eNOS expressed in baculovirus infected insect Sf9 cells assessed as conversion of [3H]-L-arginine to [3H]-L-citrullineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Q52Q3NPubMed
TargetNitric oxide synthase, endothelial(Homo sapiens (Human))
NeurAxon Inc.

Curated by ChEMBL
LigandPNGBDBM106710(CHEMBL1957357 | US8586620, 75)copy SMILEScopy InChI
Affinity DataIC50: 3.61E+4nMAssay Description:Enzyme assay using recombinant human inducible NOS (iNOS), human endothelial constitutive NOS (eNOS) or human neuronal constitutive NOS (nNOS).More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2348J0KUS Patent