Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50105470((S)-6-Amino-2-((R)-3-(1H-indol-3-yl)-2-{[4-(4-meth...)copy SMILEScopy InChI
Affinity DataIC50: 4.40nMAssay Description:Inhibitory concentration of the compound towards binding of sst2 receptor using [125I]-somatostatin as radioligand in Neuro2A cellsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8D5SPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50105470((S)-6-Amino-2-((R)-3-(1H-indol-3-yl)-2-{[4-(4-meth...)copy SMILEScopy InChI
Affinity DataIC50: 67nMAssay Description:Antagonistic activity of the compound towards sst2 receptor in GH4C1 cells a concentration of 1-2 x 10e6/mL incubated for 20 minutesMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2JW8D5SPubMed