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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Pfizer Inc
Curated by
ChEMBL
Ligand
BDBM50105470
((S)-6-Amino-2-((R)-3-(1H-indol-3-yl)-2-{[4-(4-meth...)
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Affinity Data
IC50: 4.40nM
Assay Description:
Inhibitory concentration of the compound towards binding of sst2 receptor using [125I]-somatostatin as radioligand in Neuro2A cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2JW8D5S
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Pfizer Inc
Curated by
ChEMBL
Ligand
BDBM50105470
((S)-6-Amino-2-((R)-3-(1H-indol-3-yl)-2-{[4-(4-meth...)
copy SMILES
copy InChI
Affinity Data
IC50: 67nM
Assay Description:
Antagonistic activity of the compound towards sst2 receptor in GH4C1 cells a concentration of 1-2 x 10e6/mL incubated for 20 minutes
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2JW8D5S
PubMed