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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
Dr. Karl Thomae GmbH
Curated by
ChEMBL
Ligand
BDBM50043863
(((E)-3-Pyridin-3-yl-3-{4-[2-(toluene-4-sulfonylami...)
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Affinity Data
IC50: 3.00E+3nM
Assay Description:
Displacement of the high affinity radiolabeled ligand [3H]- SQ-29,548 from the PGH-2/TXA-2 receptor in human gel-filtered platelets.
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2SB44T4
PubMed
Target
Thromboxane-A synthase
(Homo sapiens (Human))
Dr. Karl Thomae GmbH
Curated by
ChEMBL
Ligand
BDBM50043863
(((E)-3-Pyridin-3-yl-3-{4-[2-(toluene-4-sulfonylami...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.50E+4nM
Assay Description:
Inhibition test of thromboxane A2 synthetase in human gel-filtered platelets.
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2SB44T4
PubMed