Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 9 hits in this display   

LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 880nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 920nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 4.00E+3nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMitogen-activated protein kinase 1(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 1.10E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMitogen-activated protein kinase 7(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 1.20E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMAP kinase-activated protein kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 1.50E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMitogen-activated protein kinase 6(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 2.10E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMAP kinase-activated protein kinase 5(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 2.70E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent
TargetMAP kinase-activated protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM558850(US11370770, Compound 6b)copy SMILES
Affinity DataIC50: 2.70E+4nMAssay Description:Kinase activity of recombinant active full-length human MEK4 (Carna Biosciences) was measured using the ADP-Glo assay (Promega) with 3 μM recomb...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2HX1GWDUS Patent