Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065127(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)copy SMILEScopy InChI
Affinity DataIC50: 4nMAssay Description:Inhibition of [3H]-AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SF2VJHPubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065127(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)copy SMILEScopy InChI
Affinity DataIC50: 4.10nMAssay Description:Displacement of [3H]-AVP from vasopressin V2 receptor of rat kidney medulla.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC0ZT5PubMed
TargetVasopressin V1a receptor(RAT)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065127(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Inhibition of [3H]-AVP binding to Dawley rat hepatic vasopressin V1a receptor.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2SF2VJHPubMed
TargetVasopressin V1a receptor(RAT)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50065127(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)copy SMILEScopy InChI
Affinity DataIC50: 38nMAssay Description:Displacement of (Phe-3,4,5-H) Vasopressin from V1a recptor from rat liver membranes.More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC0ZT5PubMed