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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Vasopressin V2 receptor
(Rattus norvegicus (Rat))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50065127
(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)
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copy InChI
Affinity Data
IC50: 4nM
Assay Description:
Inhibition of [3H]-AVP binding to Dawley rat kidney medullary vasopressin V2 receptor.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2SF2VJH
PubMed
Target
Vasopressin V2 receptor
(Rattus norvegicus (Rat))
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50065127
(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)
copy SMILES
copy InChI
Affinity Data
IC50: 4.10nM
Assay Description:
Displacement of [3H]-AVP from vasopressin V2 receptor of rat kidney medulla.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CC0ZT5
PubMed
Target
Vasopressin V1a receptor
(RAT)
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50065127
(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)
copy SMILES
copy InChI
Affinity Data
IC50: 38nM
Assay Description:
Inhibition of [3H]-AVP binding to Dawley rat hepatic vasopressin V1a receptor.
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2SF2VJH
PubMed
Target
Vasopressin V1a receptor
(RAT)
Wyeth Research
Curated by
ChEMBL
Ligand
BDBM50065127
(CHEMBL71797 | N-[4-(5H,11H-Benzo[e]pyrrolo[1,2-a][...)
copy SMILES
copy InChI
Affinity Data
IC50: 38nM
Assay Description:
Displacement of (Phe-3,4,5-H) Vasopressin from V1a recptor from rat liver membranes.
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CC0ZT5
PubMed