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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
Astellas Pharma Inc.
Ligand
BDBM35675
(5H-1-benzazepin-5-ylidene acetamide, 1c)
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Affinity Data
Ki: 15nM ΔG°: -44.7kJ/mole
T: 2°C
Assay Description:
Chinese hamster ovary (CHO) cells stably expressing human V1a receptors. Cells were washed with phosphate buffered saline, and then collected in ice-...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q24T6GQM
PubMed
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
Astellas Pharma Inc.
Ligand
BDBM35675
(5H-1-benzazepin-5-ylidene acetamide, 1c)
copy SMILES
copy InChI
Affinity Data
Ki: 20nM ΔG°: -43.6kJ/mole
pH: 7.4 T: 2°C
Assay Description:
The affinities of test compounds for human V2 receptor were evaluated by the radioligand binding study using membrane fractions isolated from CHO cel...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q24T6GQM
PubMed