Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM572242(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)copy SMILES
BDBM572242(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)copy SMILES
Ki: 0.0540nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572242(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)copy SMILES
Ki: 100nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair
BDBM572242(2-[4-[(6S)-1,8-diazaspiro[5.5]undecan-8-yl]-1H- py...)copy SMILES
Ki: 203nMAssay Description:MRCKα, MRCKβ, ROCK1 and ROCK2 assays were performed using an IMAP fluorescence polarization assay format (Molecular Devices Inc.). 8-12 nM ...More data for this Ligand-Target Pair