Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSerine/threonine-protein kinase haspin(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL

LigandBDBM50379517(CHEMBL2012570)copy SMILEScopy InChI

Affinity DataIC50: 500nMAssay Description:Inhibition of human recombinant N-terminal MBP-tagged haspin kinase expressed in Escherichia coli DE3 after 10 mins by TR-FRET assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K29KKPubMed

TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL

LigandBDBM50379517(CHEMBL2012570)copy SMILEScopy InChI

Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of human N-terminal GST-tagged DYRK2 expressed in baculovirus using DYRKtide-F as substrate assessed as inhibition of [33P] incorporation ...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20K29KKPubMed