Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))TBA
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 149nMAssay Description:Inhibition of human TTBK1 (1 to 479 residues) using Casein as substrate measured after 40 mins in presence of [gamma33P]ATP by scintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of full length recombinant human IKKepsilon using casein as substrate incubated for 40 mins in presence of [gamma-33P-ATP] by radiometric ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))TBA
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 7.46E+3nMAssay Description:Displacement of tracer K5 from NLuc fused TBK1 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K9 from NLuc fused MARK3 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))TBA
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K9 from NLuc fused DRAK1 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed
TargetMAP/microtubule affinity-regulating kinase 4(Homo sapiens (Human))TBA
LigandPNGBDBM50585196(CHEMBL5084750)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Displacement of tracer K5 from NLuc fused MARK4 (unknown origin) expressed in HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27S7SNDPubMed