Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50461320(CHEMBL4227666)copy SMILEScopy InChI
Affinity DataIC50: 640nMAssay Description:Inhibition of GRK2 (unknown origin) preincubated for 10 mins followed by peptide substrate and ATP addition measured after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z1868PubMed
TargetG protein-coupled receptor kinase 5(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50461320(CHEMBL4227666)copy SMILEScopy InChI
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of GRK5 (unknown origin) preincubated for 10 mins followed by peptide substrate and ATP addition measured after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z1868PubMed
TargetRhodopsin kinase GRK1(Homo sapiens (Human))
University of Michigan

Curated by ChEMBL
LigandPNGBDBM50461320(CHEMBL4227666)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of GRK1 (unknown origin) preincubated for 10 mins followed by peptide substrate and ATP addition measured after 1 hr by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z1868PubMed