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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
12
hits in this display
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
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Affinity Data
Ki: 200nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
Ki: 1.50E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
Ki: 4.50E+3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
Royal Danish School of Pharmacy
Curated by
PDSP K
i
Database
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2MW2FNT
PubMed
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu1-alpha
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed
Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu6
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Compound was evaluated for agonistic activity against mGluR2 alpha metabotropic receptor subtype in rat cortical slice model
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27P8XJ2
PubMed
Target
Metabotropic glutamate receptor 4
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Compound was evaluated for agonistic activity against mGluR4a alpha metabotropic receptor subtype in rat cortical slice model
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27P8XJ2
PubMed
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonist activityof the compound at Metabotropic Excitatory Amino acid Receptors Expressed in CHO cells. mGlu2
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed
Target
Metabotropic glutamate receptor 1
(RAT)
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM50004852
(AMAA | Amino-(3-hydroxy-5-methyl-isoxazol-4-yl)-ac...)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Compound was evaluated for agonistic activity against mGluR1 alpha metabotropic receptor subtype in rat cortical slice model
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q27P8XJ2
PubMed