Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetSomatostatin receptor type 4(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068041(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)copy SMILEScopy InChI
Affinity DataKi:  1.50E+4nMAssay Description:In vitro binding affinity at somatostatin receptor 4 in transfected BHK cells using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4RNGPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Northeast Louisiana University

Curated by ChEMBL
LigandPNGBDBM50068041(1-{2-[(5-Bromo-pyridin-2-yl)-(3,4-dichloro-benzyl)...)copy SMILEScopy InChI
Affinity DataKi: >3.00E+5nMAssay Description:In vitro binding affinity at somatostatin 2 receptor in transfected HEK 293 cell using [125 I]Tyr11-SRIF-14 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TT4RNGPubMed