Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
TBA
Ligand
BDBM523771
(US11136312, Compound AH-1-33)
copy SMILES
Affinity Data
Ki: 92.8nM
Assay Description:
Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2DB851B
US Patent
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
TBA
Ligand
BDBM523771
(US11136312, Compound AH-1-33)
copy SMILES
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2DB851B
US Patent
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
TBA
Ligand
BDBM523771
(US11136312, Compound AH-1-33)
copy SMILES
Affinity Data
EC50: 130nM
Assay Description:
Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2DB851B
US Patent