Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  40.4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 1(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  3.17E+3nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 1(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  3.17E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  6.99E+3nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi:  6.99E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 5(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent
TargetSomatostatin receptor type 4(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataEC50:  21nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21C21X0PubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))TBA
LigandPNGBDBM523744(US11136312, Compound SM-I-60)copy SMILES
Affinity DataEC50:  21.3nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2DB851BUS Patent