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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Sodium- and chloride-dependent glycine transporter 1
(Homo sapiens (Human))
AbbVie Inc.
Curated by
ChEMBL
Ligand
BDBM308854
(N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imid...)
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Affinity Data
Ki: 8nM
Assay Description:
Inhibition of [3H]N-Methyl-SSR504734 binding to human recombinant GlyT1c expressed in CHO cell membranes incubated for 1 hr by liquid scintillation s...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2CC137K
PubMed
Target
Alpha-1,3-mannosyl-glycoprotein 2-beta-N-acetylglucosaminyltransferase
(Homo sapiens (Human))
AbbVie Inc.; AbbVie Deutschland GmbH & Co. KG
US Patent
Ligand
BDBM308854
(N-{(3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imid...)
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copy InChI
Affinity Data
Ki: <10nM
Assay Description:
Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2Z60R48
US Patent