Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Vasopressin V1a receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM526851
(US11186577, Cmpd. No. 105)
copy SMILES
Affinity Data
IC50: 100nM
Assay Description:
The purpose of this assay was to determine the inhibitory effect of synthesized compounds on the Vasopressin V1a receptor. The assay as performed in ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2T72MN6
US Patent
Target
Oxytocin receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM526851
(US11186577, Cmpd. No. 105)
copy SMILES
Affinity Data
IC50: 300nM
Assay Description:
This assay was performed in CHEM-1 cells expressing the human Oxytocin Receptor (hOTR) to determine the inhibitory effect of the compounds of the inv...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2T72MN6
US Patent
Target
Vasopressin V2 receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM526851
(US11186577, Cmpd. No. 105)
copy SMILES
Affinity Data
IC50: 1.00E+3nM
Assay Description:
The purpose of the assay was to determine the inhibitory effect of synthesized compounds on the Vasopressin receptor 2. The assay was performed in co...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2T72MN6
US Patent
Target
Vasopressin V1b receptor
(Homo sapiens (Human))
TBA
Ligand
BDBM526851
(US11186577, Cmpd. No. 105)
copy SMILES
Affinity Data
IC50: 1.00E+3nM
Assay Description:
The purpose of the assay is to determine the inhibitory effect of synthesized compounds on the Vasopressin V1b receptor. The assay was performed in C...
More data for this Ligand-Target Pair
Target Info
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2T72MN6
US Patent