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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
7
hits in this display
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
CIBA-GEIGY Corporation
Curated by
PDSP K
i
Database
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
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Affinity Data
Ki: 800nM
More data for this Ligand-Target Pair
Target Info
PDB
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MCE
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2Z036NF
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
CIBA-GEIGY Corporation
Curated by
PDSP K
i
Database
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
copy SMILES
copy InChI
Affinity Data
Ki: 900nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
DrugBank
MCE
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2Z036NF
PubMed
Target
Glutamate receptor ionotropic, NMDA 1
(RAT)
CIBA-GEIGY Corporation
Curated by
PDSP K
i
Database
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
Purchase
CHEMBL
DrugBank
MCE
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W094FK
PubMed
Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
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copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonistic activity at mGlu1-alpha receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
DrugBank
MCE
KEGG
MMDB
PC cid
PC sid
PDB
Patents
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
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copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonistic activity at mGlu2 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
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CHEMBL
DrugBank
MCE
KEGG
MMDB
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed
Target
Glutamate transporter homolog
(Pyrococcus horikoshii (strain ATCC 700860 / DSM 12...)
Columbia University
Curated by
ChEMBL
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
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copy InChI
Affinity Data
Kd: 10nM
Assay Description:
Binding affinity to Pyrococcus horikoshii sodium-coupled aspartate transporter L130W mutant fluorescence-based assay in presence of NaCl
More data for this Ligand-Target Pair
Target Info
PDB
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Ligand Info
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CHEMBL
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MCE
KEGG
MMDB
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In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q29C716Z
PubMed
Target
Metabotropic glutamate receptor 6
(Homo sapiens (Human))
Royal Danish School of Pharmacy
Curated by
ChEMBL
Ligand
BDBM31174
(CHEMBL29757 | D-Aspartate | D-Aspartic Acid)
copy SMILES
copy InChI
Affinity Data
EC50: >1.00E+6nM
Assay Description:
Agonistic activity at mGlu6 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
DrugBank
MCE
KEGG
MMDB
PC cid
PC sid
PDB
Patents
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2M909BH
PubMed