Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMelanocortin receptor 5(Mus musculus (Mouse))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50232419(CHEMBL4060767)copy SMILEScopy InChI
Affinity DataEC50:  6.00E+3nMAssay Description:Agonist activity at mouse MC5R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50232419(CHEMBL4060767)copy SMILEScopy InChI
Affinity DataEC50:  900nMAssay Description:Agonist activity at mouse MC1R expressed in HEK293 cells assessed as increase in forskolin-induced cAMP accumulation preincubated for 2 hrs followed ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R213MTPubMed