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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Somatostatin receptor type 3
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50099173
(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
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Affinity Data
Ki: 200nM
Assay Description:
Inhibition of human sst3 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2D50NHN
PubMed
Target
Somatostatin receptor type 1
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50099173
(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
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copy InChI
Affinity Data
Ki: 1.55E+3nM
Assay Description:
Inhibition of human sst1 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2D50NHN
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50099173
(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
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copy InChI
Affinity Data
Ki: 2.25E+3nM
Assay Description:
Inhibition of human sst5 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2D50NHN
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50099173
(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
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copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of human sst2 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2D50NHN
PubMed
Target
Somatostatin receptor type 4
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50099173
(2,4-Difluoro-N-[(R)-2-(1H-indol-3-yl)-1-(4-phenyl-...)
copy SMILES
copy InChI
Affinity Data
Ki: >1.00E+4nM
Assay Description:
Inhibition of human sst4 receptor expressed in CHO cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2D50NHN
PubMed