Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
H. Lee Moffitt Cancer Center& Research Institute

Curated by ChEMBL
LigandPNGBDBM50358561(CHEMBL1923664)copy SMILEScopy InChI
Affinity DataKi:  0.240nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC1 receptor expressed in human HCT116 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G1618KPubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
H. Lee Moffitt Cancer Center& Research Institute

Curated by ChEMBL
LigandPNGBDBM50358561(CHEMBL1923664)copy SMILEScopy InChI
Affinity DataKi:  46nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC5 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G1618KPubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
H. Lee Moffitt Cancer Center& Research Institute

Curated by ChEMBL
LigandPNGBDBM50358561(CHEMBL1923664)copy SMILEScopy InChI
Affinity DataKi:  254nMAssay Description:Displacement of Eu-NDP-alphaMSH from human MC4 receptor expressed in human HEK293 cells after 1.5 hrs by time-resolved fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2G1618KPubMed