Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGluR2 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 6(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  6.01E+3nMAssay Description:Agonist activity at rat mGluR6 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 7(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at rat mGluR7 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 8(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at rat mGluR8 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50387817(CHEMBL2058378)copy SMILEScopy InChI
Affinity DataEC50:  340nMAssay Description:Agonist activity at rat mGlu4 receptor expressed in HEK293 cells coexpressing Gq/Gi and EAAC1 assessed as intracellular calcium production measured e...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2Q2WPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  1.13E+4nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  100nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  120nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Univ. Rouen

Curated by ChEMBL
LigandPNGBDBM50088290(CHEMBL3427499)copy SMILEScopy InChI
Affinity DataEC50:  300nMAssay Description:Agonist activity at rat mGluR4 expressed in HEK293 cells assessed as induction of inositol phosphate production by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21Z464CPubMed