Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSomatostatin receptor type 5(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254243((5S)-6-(benzylamino)-6-oxo-5-[(4R)-3-oxo-4-[(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 3.40nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst5 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6D3BPubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254243((5S)-6-(benzylamino)-6-oxo-5-[(4R)-3-oxo-4-[(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 8.10nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst4 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6D3BPubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254243((5S)-6-(benzylamino)-6-oxo-5-[(4R)-3-oxo-4-[(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst2 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6D3BPubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254243((5S)-6-(benzylamino)-6-oxo-5-[(4R)-3-oxo-4-[(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 54nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst1 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6D3BPubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Vrije Universiteit Brussel

Curated by ChEMBL
LigandPNGBDBM50254243((5S)-6-(benzylamino)-6-oxo-5-[(4R)-3-oxo-4-[(3-phe...)copy SMILEScopy InChI
Affinity DataIC50: 153nMAssay Description:Displacement of [125I]-[Leu8, DTrp22, Tyr25]-somatostatin-28 from human recombinant sst3 receptor expressed in chinese hamster CCL39 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6D3BPubMed