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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Melanocyte-stimulating hormone receptor
(Mus musculus)
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217759
(CHEMBL237694 | N-(5-aminopentyl)-N-(benzo[d][1,3]d...)
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Affinity Data
Ki: 5.50E+3nM
Assay Description:
Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cells
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2X066Q5
PubMed
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217759
(CHEMBL237694 | N-(5-aminopentyl)-N-(benzo[d][1,3]d...)
copy SMILES
copy InChI
Affinity Data
Ki: 1.20E+4nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC4 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2X066Q5
PubMed
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217759
(CHEMBL237694 | N-(5-aminopentyl)-N-(benzo[d][1,3]d...)
copy SMILES
copy InChI
Affinity Data
Ki: 2.30E+4nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2X066Q5
PubMed
Target
Melanocortin receptor 3
(Homo sapiens (Human))
Uppsala University
Curated by
ChEMBL
Ligand
BDBM50217759
(CHEMBL237694 | N-(5-aminopentyl)-N-(benzo[d][1,3]d...)
copy SMILES
copy InChI
Affinity Data
Ki: 3.80E+4nM
Assay Description:
Displacement of [125I]NDP-MSH from human recombinant MC3 receptor expressed in Sf9 cells
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2X066Q5
PubMed